METABOLIC PATHWAYS, METABOLOMICS & METABONOMICS

THE PHYSIOME



However clear each gene and the amino acid sequence of its associated protein may become, it is hard to infer physiological function, from gene and/or protein, resulting in failure to solve the puzzles of (human) physiological functions (after F. Kajiya).

Lessons from genome-wide analysis of Metabolic Pathways

 Metabolic Pathways are:

1.    Plastic and species - specific

2.    Highly versatile, in a single species and in multi-genome comparisons

Examples:

1. The Citric Acid Cycle

Huynen, MA, Dandekar T and Bork, P.  Variation and evolution of the citric acid cycle: a genomic perspective. Trends in Microbiology (1999) 7, 281-291

2.  Glycolytic Pathways

Dandekar T et al. Pathway alignment: application to the comparative analysis of glycolytic enzymes. Biochem J. (1999) 343, 115-124

3.  Evolution of Metabolic pathways

Forst CV and Schulten K.  Evolution of Metabolisms: A New Method for the Comparison of Metabolic Pathways Using Genomic Information. J.Comput. Biol. (1999) 6, 343-360

3.  Concept of Elementary Flux Modes, minimal sets of steps/enzymes that could in principle operate independently of any others, for analysis of metabolic networks.

Schuster S. et al. Nature Biotech. (2000) 18, 326 - 332.

Abstract:

The concept of 'elementary flux modes' provides a mathematical tool to define and comprehensively describe all metabolic routes that are both stoichiometrically and thermodynamically feasible for a group of enzymes. We have used this concept to analyze the interplay between the pentose phosphate pathway (PPP) and glycolysis. The set of elementary modes for this system involves conventional glycolysis, a futile cycle, all the modes of PPP function described in biochemistry textbooks, and additional modes that are a priori equally entitled to pathway status. Applications include maximizing product yield in amino acid and antibiotic synthesis, reconstruction and consistency checks of metabolism from genome data, analysis of enzyme deficiencies, and drug target identification in metabolic networks.
 

Relevant Databases and Websites
 

Metabolic Pathways:
 

      BioCyc - collection of Pathway/Genome Databases

      PATHWAY at KEGG at GenomeNet

    GeneNetworks: 41 different cellular networks blending biochemical networks and signalling

     WIT - Metabolic Reconstruction

     Metalgen - Genes and Metabolism (under construction)

     Boehringer Mannheim - Biochemical Pathways

     UM-BBD - Microbial Biocatalysis/Biodegradation

    EPA Computational Toxicology website

      Reactome - a database of individual biochemical reactions from humans and non-human systems such as rat, mouse, pufferfish, and                       zebrafish,  obtained either via a literature citation or an electronic inference based on sequence similarity.

METABONOMICS


The study of metabolic responses to drugs, environmental changes and diseases. Metabonomics is an extension of

genomics (concerned with DNA) and proteomics (concerned with proteins). Following on the heels of genomics and proteomics,

metabonomics may lead to more efficient drug discovery and individualized patient treatment with drugs, among other things.

In more technical (and wordy) terms, metabonomics is the quantitative measurement of the dynamic multiparametric metabolic response of

living systems to pathophysiological stimuli or genetic modification. (Medicine.Net)

METABOLOMICS


The global study of all the small molecules produced by metabolism in an organism.

Metabolomic analysis enables the biochemical consequences of genetic variations, mutations and changes in the environment and treatment with drugs to be observed directly.

This may help in the diagnosis of disease, and development of new drugs. It may also help us to understand how environmental agents and drugs work, interact and cause side effects.

The Metabolomics Society

THE PHYSIOME PROJECT
 


Physiome Project



The Physiome Project consists of two main parts (i) the databasing of biological information and (ii) systematic approach obtaining the schema of interaction, quantitative description of interrelationship and modelling.

The idea:

The Physiome Project is a loosely integrated multi-centric program to design, develop, implement, test and document, archive and disseminate qualitative and quantitative information, databases and models of the functional behaviour of organelles, cells, tissues, organs, and organisms. It is a successor to the Genome Project. The focus of the Human Physiome Project is on the human organism, its physiology and pathophysiology, to eventually provide full working models of physiological systems that integrate the
observations from many laboratories into quantitative, self-consistent, comprehensive descriptions.

The goal is to provide to the community of scientists, physicians, teachers, and manufacturers functional descriptions of human biological systems in health and disease. A major feature of the project is the databasing of observations on all organisms for retrieval and evaluation. A network of Physiome Centres would comprise an adaptable international resource for integrated physiological systems, structured for accessibility via the Internet, for the immense databases of information on methods, data and models.

The plan

    There is a growing effort to raise consciousness about integrative biology and to provide a setting for
the results that are flowing out of laboratories concerned with genomics. molecular and cell biology, and medicine and biology in general. For those with a primary interest in therapeutics, the Physiome Project can provide a framework for determining the effects of pharmaceutical or genetic interventions on target
molecules and functional systems through a deep, comprehensive understanding of biology at the level of the cell, the tissue, the organ and the organism. The Project will need to be supported by the development of databases that follow upon those developed from the Genome and the Proteome. Physiological modelling may be considered to include the dynamics of protein folding, molecular dynamics in general,
protein-protein interactions of all sorts, from solutes in competition for binding sites on enzymes and receptors to antigen-antibody reactions. Integration at the more structured levels, organelles, cells, and broader, may not always be based on (reductionist) approaches, but will often have to be explained at molecular level as well as at the system level.

MATHEMATICAL MODELLING OF METABOLIC NETWORKS
 

Lectures in Harvard Biophysics 101 Lecture Course:

    Metabolic network flux models: Introduction to the basic concepts and linear optimization

    Metabolic network flux models: Scientific and practical use

Cascante et al., (2002) Metabolic control analysis in drug discovery and disease. Nature Biotech. 20, 243-9.